Syntheses of Pyrazole Derivatives. VI
نویسندگان
چکیده
منابع مشابه
Syntheses of Anisomycin Derivatives
The structure of anisomycin has been determined by X-ray investigation4 and the absolute configuration was confirmed by chemical correlation.5 Anisomycin has attracted considerable synthetic interest, and several synthetic studies, derivative syntheses as well as total syntheses, have been reported.6 Especially, the synthesis of its analogues has revealed the structure-activity relationship of ...
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Several new pyrazole derivatives have demonstrated promising antiproliferative and cytotoxic effects, but their poor solubility raised concerns over possible biopharmaceutical limitations. In order to improve their pharmaceutical potential we performed the biopharmaceutical profiling for nine pyrazole compounds using in vitro and computational methods. The experimental solubility was determined...
متن کاملPyrazole Carbohydrazide Derivatives of Pharmaceutical Interest
The main purpose of this paper is to provide an insight into the biological activities of pyrazole derivatives which contain the carbohydrazide moiety.
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ژورنال
عنوان ژورنال: YAKUGAKU ZASSHI
سال: 1963
ISSN: 0031-6903,1347-5231
DOI: 10.1248/yakushi1947.83.8_745